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Put two entries side by side — evidence, mechanism, risks, and community claims.

AICAR

Preclinical
Banned in sport
Summary
Cell-permeable AMPK-activating nucleoside analog famously studied as an exercise mimetic in sedentary mice; WADA-prohibited.
Categories
Metabolic & Body Comp, Performance
Mechanism
Converted to ZMP which mimics AMP, activating AMPK and PGC-1α metabolic gene programs favoring an oxidative phenotype.
Half-life
Hours
Routes
Subcutaneous injection; Intravenous
Legal / access
WADA prohibited. Not an approved exercise drug. Research chemical only.
Key risks
  • Lactic acidosis risk theoretical
  • Uric acid changes
  • Unknown chronic toxicity at performance doses
Common claims
  • Cardio in a bottle narratives
  • Fat oxidation
  • Endurance without training (overstated)
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